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Synthesis of 2-R-2-(1-Aryl-7,8-Dimethoxy-5H-2,3-Benzodiazepin-4-yl)Acetic Acid Esters in the Eschenmoser Reaction

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Chemistry of Heterocyclic Compounds Aims and scope

A method for the synthesis of 2-R-2-(1-aryl-7,8-dimethoxy-5H-2,3-benzodiazepin-4-yl)acetic acid esters from 2-R-2-(1-aryl-7,8-dimethoxy-5H-2,3-benzodiazepin-4-ylsulfanyl)acetic acid esters through Eschenmoser reaction has been developed.

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Authors and Affiliations

  1. L. M. Litvinenko Institute of Physical Organic Chemistry and Coal Chemistry, National Academy of Sciences of Ukraine, 70 R. Luxemburg St., Donetsk, 83114, Ukraine

    E. S. Sizonenko, V. Yu. Popov, S. Yu. Suikov & S. L. Bogza

  2. I. M. Gubkin Russian State University of Oil and Gas, 65 Leninsky Ave., Moscow, 119991, Russia

    I. K. Kobrakov

Authors
  1. E. S. Sizonenko
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  2. I. K. Kobrakov
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  3. V. Yu. Popov
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  4. S. Yu. Suikov
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  5. S. L. Bogza
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Corresponding author

Correspondence to E. S. Sizonenko.

Additional information

Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 9, pp. 1451-1456, September, 2013.

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Sizonenko, E.S., Kobrakov, I.K., Popov, V.Y. et al. Synthesis of 2-R-2-(1-Aryl-7,8-Dimethoxy-5H-2,3-Benzodiazepin-4-yl)Acetic Acid Esters in the Eschenmoser Reaction. Chem Heterocycl Comp 49, 1352–1357 (2013). https://doi.org/10.1007/s10593-013-1384-0

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  • DOI: https://doi.org/10.1007/s10593-013-1384-0

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