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Dichloroacetylaroylmethanes as two-carbon synthons in the Biginelli reaction

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

Acid-catalyzed cyclocondensation in a three component system of dichloromethylacetylbenzoylmethanes, urea, and aromatic aldehydes occurred regio-and stereoselectively to give polyfunctional derivatives of perhydropyrimidine.

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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 9, 1414–1417, September, 2006.

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Mamedov, V.A., Mustakimova, L.V., Gubaidullin, A.T. et al. Dichloroacetylaroylmethanes as two-carbon synthons in the Biginelli reaction. Chem Heterocycl Compd 42, 1229–1232 (2006). https://doi.org/10.1007/s10593-006-0230-z

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  • DOI: https://doi.org/10.1007/s10593-006-0230-z

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