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Activated nitriles in heterocyclic synthesis novel synthesis of thiadiazolo[2,3-a]pyridine derivatives

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Abstract

Several new thiadiazolo[2,3-a]pyridine, thiazole and coumarin derivatives were synthesized via the reaction of 2-cyanomethylthiadiazole with cinnamonitrile, mercaptoacetic acid and salicylaldehyde.

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Authors and Affiliations

  1. Chemistry Department, Faculty of Science, Damietta-Mansoura University, Egypt

    Salah Zaki Ahmed Sowellim, Mohamed Nabil Mohamed Khodeir, Ahmed Ibrahim Osman & Abdel Ghani Ali Elagamey

Authors
  1. Salah Zaki Ahmed Sowellim
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  2. Mohamed Nabil Mohamed Khodeir
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  3. Ahmed Ibrahim Osman
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  4. Abdel Ghani Ali Elagamey
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Ahmed Sowellim, S.Z., Mohamed Khodeir, M.N., Osman, A.I. et al. Activated nitriles in heterocyclic synthesis novel synthesis of thiadiazolo[2,3-a]pyridine derivatives. Arch. Pharm. Res. 11, 253–256 (1988). https://doi.org/10.1007/BF02857757

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  • DOI: https://doi.org/10.1007/BF02857757

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