Abstract
In order to search target organs and to study the mechanism of the action of steroids with separated biological functions, tritium-labeled pregna-d'-pentaranes were synthesized by an original procedure, and their interaction with a progesterone receptor was investigated. The uterine progesterone receptor was shown to be the only specific binding protein for these compounds.
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Translated fromIzvestiya Akademii Nauk. Seriya Khimicheskaya, No. 8, pp. 1532–1535, August, 1997.
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Kamernitsky, A.V., Levina, I.S., Kulikova, L.E. et al. Synthesis of [3H]-cycloalkanoprogesterones (pregna-d'-pentaranes) and study of their interaction with a progesterone receptor. Russ Chem Bull 46, 1468–1471 (1997). https://doi.org/10.1007/BF02505688
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DOI: https://doi.org/10.1007/BF02505688