Abstract
8-Substituted tetrahydropyrido[3,2-e]pyrrolizines are formed in the [3+2]-cycloaddition of 2-formyltetrahydropyrrolo[3,2-c]pyridine and acrolein, acrylonitrile, and methyl acrylate in the presence of trilon B.
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Additional information
Russian International Friendship University, 117923 Moscow. Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 12, pp. 1670–1675, December, 1998.
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Varlamov, A.V., Borisova, T.N., Barge, S.B. et al. Unusual [3+2]-cycloaddition of acrylic acid derivatives to 7-formyl-4,5,6,7-tetrahydro-4,5,7-trimethylpyrrolo[3,2-c]pyridine under Michael reaction conditions. Chem Heterocycl Compd 34, 1418–1422 (1998). https://doi.org/10.1007/BF02317813
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DOI: https://doi.org/10.1007/BF02317813