Abstract
We have shown that heterocyclization of N-tosyl- and N-acetyl derivatives of 8-(allylamino)quinoline with iodine occurs with formation of 3-iodomethyl-1-p-toluenesulfonyl-2,3-dihydropyrazino[3,2,1-i,j]quinolinium and 1-acetyl-3-iodomethyl-2,3-dihydropyrazino[3,2,1-i,j]quinolinium iodides.
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Additional information
Chelyabinsk State University, Chelyabinsk 454136. Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 6, pp. 781–784, June, 1997.
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Vorob'ev, D.V., Tikhonova, Y.V., Kim, D.G. et al. Synthesis and heterocyclization of allyl derivatives of 8-aminoquinoline. Chem Heterocycl Compd 33, 680–683 (1997). https://doi.org/10.1007/BF02291799
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DOI: https://doi.org/10.1007/BF02291799