Experientia

, Volume 39, Issue 6, pp 591–592 | Cite as

Stereoselective binding of 4,5-dihydrodiazepam to human serum albumin

  • I. Fitos
  • M. Simonyi
Article

Summary

S(+)-4,5-dihydrodiazepam was found to have higher binding affinity for human serum albumin than its antipode. The binding of 4-carbamoyl-4,5-dihydrodiazepam is weak and not stereoselective.

Keywords

Albumin Serum Albumin Binding Affinity Human Serum Human Serum Albumin 

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Copyright information

© Birkhäuser Verlag 1983

Authors and Affiliations

  • I. Fitos
    • 1
  • M. Simonyi
    • 1
  1. 1.Central Research Institute for Chemistry of The Hungarian Academy of SciencesBudapestHungary

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