Summary
From the unripe fruits ofSapium indicum, an irritant compound, sapintoxin, was isolated. Spectroscopic data together with selective hydrolysis and partial synthesis confirmed sapintoxin as 12-O-[N-methylaminobenzoyl]-13-O-acetyl-4-deoxyphorbol.
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Taylor, S.E., Gafur, M.A., Choudhury, A.K. et al. Sapintoxin A, a new biologically active nitrogen containing phorbol ester. Experientia 37, 681–682 (1981). https://doi.org/10.1007/BF01967918
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DOI: https://doi.org/10.1007/BF01967918