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Conformation and local anesthetic activity of carbanilates

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Summary

The influence of spatial configuration on intensity, onset, and duration of anesthetic effect has been observed in some carbanilate local anesthetics of fixed conformation. Synthesis of the carbanilates is described.

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Beneš, L., Štolc, S., Bauer, V. et al. Conformation and local anesthetic activity of carbanilates. Experientia 38, 1348–1349 (1982). https://doi.org/10.1007/BF01954944

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