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Chemistry of Heterocyclic Compounds

, Volume 5, Issue 1, pp 108–111 | Cite as

5-Substituted pyrimidine derivatives

II. Synthesis of 5, 6-dihydropyrrolo[2,3-d]pyrimidines (5,7-diazaindolines)
  • K. A. Chkhikvadze
  • N. I. Koretskaya
  • N. S. Rodnyanskaya
  • O. Yu. Magidson
Article
  • 38 Downloads

Abstract

The properties and reactivities of 4-hydroxy- and 2,4-dihydroxy-5-(β-hydroxyethyl)pyrimidines and of the products of their transformations have been studied. 4-Chloro- and 2,4-dichloro-5-(β-chloroethyl)pyrimidines have been obtained. A number of 4-alkyl(aryl)amino-5-(β-chloroethyl)pyrimidines have been synthesized, and they have been converted into derivatives of 5,6-dihydropyrrolo[2,3-d]pyrimidine.

Keywords

Organic Chemistry Pyrimidine Pyrimidine Derivative 
These keywords were added by machine and not by the authors. This process is experimental and the keywords may be updated as the learning algorithm improves.

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Copyright information

© Consultants Bureau 1971

Authors and Affiliations

  • K. A. Chkhikvadze
    • 1
  • N. I. Koretskaya
    • 1
  • N. S. Rodnyanskaya
    • 1
  • O. Yu. Magidson
    • 1
  1. 1.Ordzhonikidze All-Union Chemical and Pharmaceutical Scientific-Research InstituteMoscow

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