Abstract
The phosphorylation of the hydrochloride salt of S-butyl N-tert-butylaminothioacetate using phosphorus chlorides in the presence of triethylamine gave a new type of 1,3,2-oxazaphospholines with an alkylthio group at C5 in the oxazaphospholine ring.
Literature cited
Yu. G. Gololobov and Yu. V. Balitskii, Zh. Obshch. Khim.,44, No. 10, 2356 (1974).
Yu. G. Gololobov and L. I. Nesterova, Zh. Org. Khim.,14, No. 4, 739–745 (1978).
Yu. G. Gololobov and L. I. Kruglik, Zh. Org. Khim.,17, No. 4, 869 (1981).
Author information
Authors and Affiliations
Additional information
Translated from Izvestiya Akademii Nauk SSSR, Seriya Khimicheskaya, No. 7, pp. 1646–1647, July, 1990.
Rights and permissions
About this article
Cite this article
Gololobov, Y.G., Kruglik, L.I. Heterocyclization of thiol esters ofα-aminocarboxylic acids with the formation of 5-alkylthio-Δ4-1,3,2-oxazaphospholines. Russ Chem Bull 39, 1495–1496 (1990). https://doi.org/10.1007/BF00957870
Received:
Issue Date:
DOI: https://doi.org/10.1007/BF00957870