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Chemistry of Heterocyclic Compounds

, Volume 5, Issue 5, pp 674–676 | Cite as

Synthesis of 1-aryldihydro uracils and 1-aryl-2-thiodihydro uracils and their transformations

  • R. S. Baltrushis
  • I. I. Marioshyus
Article
  • 28 Downloads

Abstract

During the interaction of n-toluidine, n-anisidine, and n-phenetidine with methyl acrylate, the corresponding methyl esters of N-aryl-β-alanines and the corresponding N-aryl-β-alanines were obtained which were converted into 1-aryldihydro uracils and 1-aryl-2-thiodihydro uracils and then into 1-aryl-5-bromodehydrouracils, 1-aryl-2-thiohexahydropyrimidines, the hydrazides of N-aryl-β-alanines and 1-aryl-2-carboxymethylthio-4-oxo-1,4,5,6-tetrahydropyrimidines.

Keywords

Methyl Ester Organic Chemistry Methyl Ester Acrylate 
These keywords were added by machine and not by the authors. This process is experimental and the keywords may be updated as the learning algorithm improves.

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Copyright information

© Consultants Bureau 1972

Authors and Affiliations

  • R. S. Baltrushis
    • 1
  • I. I. Marioshyus
    • 1
  1. 1.Kaunas Polytechnic InstituteLithuania

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