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Synthesis and anticholine esterase properties of S-ethynyl esters of thiophosphoric acids

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Bulletin of the Academy of Sciences of the USSR, Division of chemical science Aims and scope

Conclusions

Introduction of acetylenic bond into the α-position of the thioester group of thiophosphoric acids leads to a sharp intensification of the ability of these compounds to inhibit choline esterase of different origins.

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Translated from Izvestiya Akademii Nauk SSSR, Seriya Khimicheskaya, No. 7, pp. 1602–1605, July, 1983.

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Godovikov, N.N., Vikhreva, L.A., Babasheva, K.K. et al. Synthesis and anticholine esterase properties of S-ethynyl esters of thiophosphoric acids. Russ Chem Bull 32, 1453–1455 (1983). https://doi.org/10.1007/BF00954356

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  • DOI: https://doi.org/10.1007/BF00954356

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