Conclusions
The direct condensation of iodoanilines with 2-methyl-3-bu1yn-2-ol gave acetylenic carbinols, whose cleavage by the reverse Favorskii reaction leads to ethynylanilines.
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Translated from Izvestiya Akademii Nauk SSSR, Seriya Khimicheskaya, No. 5, pp. 1184–1186, May, 1982.
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Bardamova, M.I., Trotsenko, Z.P. & Kotlyarevskii, I.L. Acetylenic derivatives of aniline. Russ Chem Bull 31, 1057–1059 (1982). https://doi.org/10.1007/BF00949973
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DOI: https://doi.org/10.1007/BF00949973