Abstract
2-Amino-6-aryl-imidazo(2,1-b)-1,3,4-thiadiazoles (1 a-f) were condensed with 1,3-ketocarboxylates e. g. ethyl-butyroacetate, ethyl-benzoylacetate, 4-nitrobenzoylacetate or ethyl-cyclopentanone(2)-carboxylate and ethyl-cyclohexanone(2)-carboxylate directly to imidazo(2,1-b)-1,3,4-thiadiazolo(3,2-a) pyrimidones-(6) (4 a-f, 5 a-f, 6 d, e, 7 a-f, 8 a, d).
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11. Mitt. über Heterocyclen; 10. Mitt.Paul, H., Sitte, A., Wessel, R., Arch. Pharm. (Weinheim), im Druck.
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Paul, H., Wessel, R. & Huschert, G. Zur Synthese von Imidazo(2,1-b)-1,3,4-thiadiazolo(3,2-a)-pyrimidonen-(6). Monatshefte für Chemie 112, 209–213 (1981). https://doi.org/10.1007/BF00911087
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DOI: https://doi.org/10.1007/BF00911087