Derivatives of phosphorus acids and 2-chloro-2-propen-1-ol

  • B. A. Arbuzov
  • V. M. Zoroastrova
  • N. D. Ibragimova
  • I. D. Neklesova
  • B. L. Mazur
  • M. A. Kudrina
  • N. V. Egorova
  • I. S. Iraidova
Organic Biological Chemistry
  • 18 Downloads

Conclusions

  1. 1.

    A number of derivatives of phosphorus acids and 2-chloro-2-propen-l-ol were prepared, and some of their chemical and biological properties were studied.

     
  2. 2.

    The 2-chloroallyl phosphorus derivatives synthesized are contact insecticides of low activity.

     
  3. 3.

    Fungicidal active with respect toTrichophyton gypseum and Epidermophyton increases with lengthening of the hydrocarbon chains of the alcohol residues of the phosphorus esters, whereas toxieity with respect to warm-blooded animals diminishes considerably.

     
  4. 4.

    The compounds studied have moderate activity with respect to Mycobacterium tuberculosis hominis.

     

Keywords

Alcohol Ester Phosphorus Hydrocarbon Tuberculosis 

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Literature cited

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Copyright information

© Consultants Bureau 1968

Authors and Affiliations

  • B. A. Arbuzov
    • 1
    • 2
    • 3
  • V. M. Zoroastrova
    • 1
    • 2
    • 3
  • N. D. Ibragimova
    • 1
    • 2
    • 3
  • I. D. Neklesova
    • 1
    • 2
    • 3
  • B. L. Mazur
    • 1
    • 2
    • 3
  • M. A. Kudrina
    • 1
    • 2
    • 3
  • N. V. Egorova
    • 1
    • 2
    • 3
  • I. S. Iraidova
    • 1
    • 2
    • 3
  1. 1.A. M. Butlerov Chemical InstituteV. I. Ul'yanov-Lenin Kazan' State UniversityUSSR
  2. 2.A. E. Arbuzov Institute of Organic and Physical ChemistryAcademy of Sciences of the USSRUSSR
  3. 3.Kazan' State Medical InstituteUSSR

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