Skip to main content
Log in

Methods of preparation of p-nitroacetophenone (review)

  • Methods of Synthesis and Technological Production of Medicines
  • Published:
Pharmaceutical Chemistry Journal Aims and scope

This is a preview of subscription content, log in via an institution to check access.

Access this article

Price excludes VAT (USA)
Tax calculation will be finalised during checkout.

Instant access to the full article PDF.

Institutional subscriptions

Literature cited

  1. S. G. Barashkov, Med. Promst. SSSR, No. 4, 40–43 (1963).

    Google Scholar 

  2. S. G. Barashkov, P. M. Kochergin, et al., Khim.-farm. Zh., No. 5, 55–57 (1972).

    Google Scholar 

  3. O. S. Vladyrchik, L. L. Bespalova, P. M. Kochergin, et al., Zh. Prikl. Khim.,32, 2250–2255 (1959).

    Google Scholar 

  4. O. S. Vladyrchik, L. L. Bespalova, P. M. Kochergin, et al., Zh. Prikl. Khim., 2744–2799.

  5. O. S. Vladyrchik, P. M. Kochergin, K. E. Novikova, et al., Zh. Prikl. Khim., 1830–1834.

  6. B. I. Golovanenko and B. D. Kruzhalov, Zh. Prikl. Khim., 1830–1834.

  7. N. N. Dykhanov and A. I. Roshchenko, Inventor's Certificate (USSR), No. 172, 745 (1965); Byull. Izobr., No. 14, p. 17 (1965).

  8. A. S. Elina, V, A. Mikhalev, and A. P. Skoldinov, in: Main Research Projects of the VNIKhFI (All-Union Scientific-Research Chemical-Pharmaceutical Institute): Review of Activities over the Period 1920–1957 [in Russian], Moscow (1959), pp. 338–368.

  9. M. N. Kolosov, M. M. Shemyakin, A. S. Khokhlov, et al., in: The Chemistry of Antibiotics [in Russian], Moscow (1961), Vol. 1, pp. 354–356.

    Google Scholar 

  10. A. A. Kolpachki and E. P. Babin, Methods of Preparation of Chemical Reagents and Compounds [in Russian], Moscow (1970), No. 22, pp. 135–137.

    Google Scholar 

  11. P. M. Kochergin, Zh. Obshch. Khim.,27, 3204–3207 (1957).

    Google Scholar 

  12. P. M. Kochergin, L. S. Blinova, V. M. Titkova, et al., Zh. Org. Khim.,7, 2157–2161 (1957).

    Google Scholar 

  13. P. M. Kochergin, L. S. Blinova, and R. M. Titkova, Med. Promst. SSSR, No. 10, 40–42 (1956).

    Google Scholar 

  14. P. M. Kochergin, L. S. Blinova and R. M. Titkova, Med. Promst., No. 11, 35–38.

  15. P. M. Kochergin, L. S. Blinova, R. M. Titkova, et al., in: All-Union Conference on the Chemistry of Nitro-Compounds. No. 2. Proceedings [in Russian], Moscow (1965), pp. 16–22.

    Google Scholar 

  16. P. M. Kochergin, L. S. Blinova, and R. M. Titkova, Inventor's Certificate (USSR) No. 178, 816; Byull. Izobre., No. 4, p. 20 (1966).

  17. P. M. Kochergin and K. S. Bushueva, Zh. Obshch. Khim.,32, 3030–3035 (1962).

    Google Scholar 

  18. P. M. Kochergin, O. S. Vladyrchik, and L. L. Bespalova, Inventor's Certificate (USSR) No. 119, 524; Byull. Izobr., No. 9, p. 15 (1959).

  19. P. M. Kochergin, A. A. Grigorovskii, V. A. Zasosov, et al., Inventor's Certificate (USSR) No. 110, 906; Byull. Izobre., No. 1, p. 29 (1958).

  20. P. M. Kochergin, A. M. Grigorovskii, V. A. Zasosov, et al., Inventor's Certificate. (USSR) No. 111, 768; Byull. Izobre., No. 3, p. 33.

  21. M. Ya. Kraft, K. I. Znaeva, and E. P. Sytina, Inventor's Certificate (USSR) No. 118, 214.

  22. N. N. Lebedev, The Chemistry and Technology of Major Organic and Petro-chemical Syntheses [in Russian], Moscow (1981), p. 509.

  23. M. Levi and K. Markov, Khim.-farm. Zh., No. 6, 13–15 (1969).

    Google Scholar 

  24. Sh. A. Mamedov and A. S. Agaev, Inventor's Certificate. (USSR) No. 126, 500; Izobreteniya, No. 5, p. 18 (1960).

  25. Nam Ch'ih Ir and Kuo Tia Kuon, Vestn. AN KNDR, No. 2, 37–41 (1961); Ref. Zh. Khim., 12Zh150 (1962).

    Google Scholar 

  26. E. I. Nezhuta and A. V. Savitskii, Med. Promst. SSSR, No. 4, 9–10 (1956).

    Google Scholar 

  27. E. I. Nezhuta and A. V. Savitskii, Zh. Obshch. Khim.,27, 1079–1080 (1957).

    Google Scholar 

  28. British Patent No. 804, 467 (1958); Chem. Abstr.,53, P12243I.

  29. British Patent No. 691, 386; Chem. Abstr.,48, 8825.

  30. Hungarian Pat. No. 12,892 (1977); Chem. Abstr.,87, P5616m.

  31. Hungarian Pat. No. 162,625 (1974); Ref. Zh. Khim., 6H124P (1976).

  32. East German Pat. No. 28,919 (1964); Ref. Zh. Khim., 8N150P (1965).

  33. East German Pat. No. 60,998 (1968); Ref. Zh. Khim., 20N477P (1969).

  34. East German Pat. No. 125,753 (1977); Ref. Zh. Khim., 13056P (1978).

  35. Italian Pat. No. 619,000 (1969); Chem. Abstr.,56, 7219. British Pat. No. 918,496 (1963); Ref. Zh. Khim., 3N143P (1964).

  36. Polish Pat. No. 55,219 (1968); Ref. Zh. Khim., 2N215 (1970).

  37. Polish Pat. No. 47,452 (1963); Ref. Zh. Khim., 4N80 (1965).

  38. Polish Pat. No. 47,449 (1963); Ref. Zh. Khim., 22N104P (1964).

  39. Rumanian Pat. No. 58,573 (1975). Chem. Abstr.,89, 108 671w.

  40. US Pat. No. 3,117,915 (1964); Chem. Abstr.,60, 9202f.

  41. US Pat. No. 3,280,200 (1966); Chem. Abstr.,66, P28531k.

  42. West German Pat. No. 1,172,658 (1965); Ref. Zh. Khim., 24N79P (1965).

  43. West German Pat. No. 1,212,970 (1966); Ref. Zh. Khim., 2N284P (1968).

  44. West German Pat. No. 1,119,246; Ref. Zh. Khim., 3N50P (1964).

  45. Czechoslovak Pat. No. 85,397 (1955); Chem. Abstr.,50, 10774g.

  46. Czechoslovak Pat. No. 89,196; Chem. Abstr.,54, 2263.

  47. Czechoslovak Pat. No. 146,833 (1973); Ref. Zh. Khim., 20N118P (1975).

  48. Swiss Pat. No. 305,862 (1968); Ref. Zh. Khim., 9N171 (1970).

  49. Preparative Organic Chemistry [in Russian], Moscow (1959), p. 217.

  50. A, I. Rakhimov, The Chemistry and Technology of Organic Peroxides [in Russian], Moscow (1979), pp. 40–45.

  51. M. V. Rubtsov and A. G, Baichikov, Synthetic Pharmaceutical Chemicals [in Russian], Moscow (1971), pp. 56–58.

  52. V. V. Sal'nikov, Izv. Vyssh. Uchebn. Zaved., Khiim. Khim. Tekhnol.,4, 621 (1961).

    Google Scholar 

  53. Ch. S. Shen, G. Kh. Guan, Ts. T. Yan, et al., Med. Promst., SSSR, No. 5, 36 (1958).

    Google Scholar 

  54. Al Neirabeyeh, J. C. Siegler, B. Gross, et al., Synthesis, No. 12, 811–813 (1976).

    Google Scholar 

  55. L. Amoretti and F. Mossini, Farm. Ed. Sci.,22, 796–800 (1967).

    Google Scholar 

  56. F. Arndt and B. Eistert, Chem. Ber.,61, 1118–1122 (1928).

    Google Scholar 

  57. F. Arndt, B. Eistert, and W. Ender, Chem. Ber.,62, 44–56 (1929).

    Google Scholar 

  58. J. M. A. Baas and B. M. Wepster, Recl. Trav. Chim.,91, 831–835 (1972).

    Google Scholar 

  59. F. Beilstein and A. Kuhlberg, Ann. Chem.,156, 206 (1870).

    Google Scholar 

  60. G. Biglino and G. M. Nano, Ann. Chim.,57, 1533–1549 (1967).

    Google Scholar 

  61. R. E. Bowman, J. Chem. Soc., 322–324 (1950).

  62. L. Brandt and R. Verbesset, Tetrahedron,28, 89–93 (1972).

    Google Scholar 

  63. H. C. Brown and W. H. Bonner, J. Am. Chem. Soc.,76, 605–606 (1954).

    Google Scholar 

  64. R. G. Coombes and L. W. Russel, J. Chem. Soc., Perkin Trans. II, No. 7, 830–834 (1974).

    Google Scholar 

  65. R. G. Coombes and L. W. Russel, J. Chem. Soc., Perkin Trans. I, No. 14, 1751–1752 (1974).

    Google Scholar 

  66. E. J. Corey and D. Seebach, Angew. Chem.,77, 1134, 1135 (1965).

    Google Scholar 

  67. B. Davies and C. B. Thomas, J. Chem. Soc., Perkin I, No. 1, 65–70 (1975).

    Google Scholar 

  68. G. Desseigne, Mem. Poudres, 46–47, 15–26 (1964–1965); Chem. Abstr.,66, 20673m.

    Google Scholar 

  69. R. E. Erickson, P. J. Andrulis, J. E. Collins, et al., J. Org. Chem.,34, 2961–2966 (1969).

    Google Scholar 

  70. J. Ernest and Z. Vesely, Chem. Listy,47, 746–749 (1953).

    Google Scholar 

  71. A. H. Ford-Moore and H. H. Rydon, J. Chem. Soc., 679–681 (1946).

  72. J. Grundy, J. Chem. Soc., 5087–5088.

  73. A. Hajos, Mag. Tud. Akad. Kémiai, Tud. Osztál. Közl.,12, 219–223 (1959).

    Google Scholar 

  74. C. Hanson, T. Kaghazchi, and M. W. Pratt, ACS Symp. Ser.,22, 132–155 (1976).

    Google Scholar 

  75. H. B. Hass and M. L. Bender, J. Am. Chem. Soc.,71, 3482–3485 (1949).

    Google Scholar 

  76. M. Itaya, Y. Takai, and K. Suzuki, Yakugaku Zasshi,81, 1629–1632 (1961).

    Google Scholar 

  77. H. Kaneyuki, Bull. Chem. Soc. Jpn.,35, 519–523 (1962).

    Google Scholar 

  78. H. Kaneyuki, Bull. Chem. Soc. Jpn., 523–525.

  79. T. Kameo and O. Manabe, Nippon Kagaku Kaishi, No. 1, 195–197 (1974).

    Google Scholar 

  80. M. H. Klowoen and M. Boelens, Recl. Trav. Chim.,79, 1022–1033 (1960).

    Google Scholar 

  81. Z. Kulicki, Zesz. Nauk Politech. Salaskiej,154, 23–28 (1966), Ref. Zh. Khim., 4G188 (1967).

    Google Scholar 

  82. L. M. Long and H. D. Troutman, J. Am. Chem. Soc.,71, 2473–2475 (1949).

    Google Scholar 

  83. R. Maurel, J.-M. Boquet, and J.-E. Germain, Bull. Soc. Chim. Fr., No. 3, 1012 (1966).

    Google Scholar 

  84. R. B. Merrifield, J. Am. Chem. Soc.,85, 2149 (1963).

    Google Scholar 

  85. D. Milstein and J. K. Stille, J. Am. Chem. Soc.,100, 3636–3638 (1978).

    Google Scholar 

  86. H. Nieuwenhuyse and R. Louw, Tetrahedron Lett., No. 44, 4141 (1971).

    Google Scholar 

  87. K. Ogura and G. Tsuchihashi, Tetrahedron Lett., No. 34, 3151.

  88. G. A. Olah, A. P. Fung, and S. C. Narang, J. Org. Chem.,46, 3533–3537 (1981).

    Google Scholar 

  89. G. A. Olah and H. C. Lin, J. Am. Chem. Soc.,96, 2892–2898 (1974).

    Google Scholar 

  90. G. A. Olah, S. C. Narang, and A. P. Fung, J. Org. Chem.,46, 2706–2709 (1981).

    Google Scholar 

  91. B. W. Palmer and A. Fry, J. Labelled Compounds,6, 303–304 (1970).

    Google Scholar 

  92. I. Partchamazad, M. Khosrovi, and M. Fakhrai, Compt. Rend. Acad. Sci.,C287, 373–375 (1978).

    Google Scholar 

  93. A. Patchornik, and M. Kraus, J. Am. Chem. Soc.,92, 7587–7758 (1970).

    Google Scholar 

  94. H. Paul, J. Prakt. Chem.,21, 186–197 (1963).

    Google Scholar 

  95. G. H. Posner and C. E. Whitten, Tetrahedron Lett., No. 53, 4647–4650 (1970).

    Google Scholar 

  96. H. Sagae, M. Fujihira, T. Osa, et al., Chem. Lett., No. 7, 793–796 (1977).

    Google Scholar 

  97. J. Slosar and V. Sterba, Chem. Prumysl,15, 270–272 (1965).

    Google Scholar 

  98. E. C. Sterling and M. T. Bogert, J. Org. Chem.,4, 20–28 (1939).

    Google Scholar 

  99. M. Tamura, T. Yöshida, and K. Namba, Kogyo Kagaku,29, 139–150 (1968).

    Google Scholar 

  100. P. Truitt, R. Stead, L. M. Long, et al., J. Am. Chem. Soc.,71, 3511–3513 (1949).

    Google Scholar 

  101. S. Uemura, A. Toshimitsu, and M. Okano, J. Chem. Soc., Perkin Trans. I, No. 9, 1076–1079 (1978).

    Google Scholar 

  102. H. G. Walker and C. R. Hauser, J. Chem. Soc.,68, 1386–1388 (1946).

    Google Scholar 

  103. D. Wichterie and P. Cefelin, Chem. Listy,50, 1474–1478 (1956).

    Google Scholar 

  104. T. Zdrojek, D. Zyto, and M. Ziolko, Chem. Prumysl,21, 161–163 (1971).

    Google Scholar 

Download references

Author information

Authors and Affiliations

Authors

Additional information

Translated from Khimiko-farmatsevticheskii Zhurnal, Vol. 19, No. 1, pp. 62–75, January, 1985.

Rights and permissions

Reprints and permissions

About this article

Cite this article

Erofeev, Y.V., Kochergin, P.M., Azizov, U.M. et al. Methods of preparation of p-nitroacetophenone (review). Pharm Chem J 19, 47–59 (1985). https://doi.org/10.1007/BF00767105

Download citation

  • Received:

  • Issue Date:

  • DOI: https://doi.org/10.1007/BF00767105

Keywords

Navigation