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Phthalazine and heterocycles related to it

VI. Derivatives of 4-phthalazone-1-carboxylic acids with aminoalkyl chains


The synthesis of a number of dialkylaminoalkyl esters and the corresponding amides of 4-phthalazone-1-carboxylic acids has been described. Some of these compounds possess local anaesthetic and short-term hypotensive activity.

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Translated from Khimiko-Farmatsevticheskii Zhurnal, No. 9, pp. 35–38, September, 1968.

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Grablyauskas, K.V., Rekhlyavichyus, V.Y., Grablyauskene, M.I. et al. Phthalazine and heterocycles related to it. Pharm Chem J 2, 506–509 (1968).

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  • Ester
  • Organic Chemistry
  • Amide
  • Hypotensive Activity
  • Phthalazine