Conclusions
Starting with 3-phenylpyrrolidine, we synthesized a series of aminoketones, derivatives of butyro-, valero-, and caprophenones, and quaternary spiropyrrolidines. The aminoketones showed adrenolytic and nicotinolytic activity.
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For Parts I and II see [1] and [2].
Translated from Khimiko-Farmatsevticheskii Zhurnal, No. 8, pp. 25–30, August, 1968.
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Chigarev, A.G., Ioffe, D.V. Synthesis of adrenolytic substances. Pharm Chem J 2, 435–439 (1968). https://doi.org/10.1007/BF00759395
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DOI: https://doi.org/10.1007/BF00759395