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Chemistry of Natural Compounds

, Volume 30, Issue 1, pp 116–120 | Cite as

Biochemical investigation of cholinesterases and carboxylesterases from the cotton bollwormHeliothis armigera

  • A. M. Kulieva
  • D. N. Dalimov
  • G. M. Dorenskaya
  • O. V. Charieva
  • V. I. Rozengart
  • L. I. Kugusheva
  • S. N. Moralev
  • B. N. Babaev
  • A. A. Abduvakhabov
Article

Abstract

The interaction of the esterases of the cotton bollworm Heliothis armigera with a series of OO-dialkyl S-propargyl phosphorothioates has been studied. In contrast to human and murine ACEs, the hydrophobic regions of the active surfaces of the bollworm ACEs are very feebly expressed. At the same time, the hydrophobic regions in the areas of the esterase points are broader than those of murine CBEs and are adapted for the sorption of normal radicals. These compounds are selective inhibitors of CBEs and can be used as insecticide synergists.

Keywords

Organic Chemistry Active Surface Normal Radical Cholinesterase Selective Inhibitor 
These keywords were added by machine and not by the authors. This process is experimental and the keywords may be updated as the learning algorithm improves.

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Copyright information

© Plenum Publishing Corporation 1994

Authors and Affiliations

  • A. M. Kulieva
  • D. N. Dalimov
  • G. M. Dorenskaya
  • O. V. Charieva
  • V. I. Rozengart
  • L. I. Kugusheva
  • S. N. Moralev
  • B. N. Babaev
  • A. A. Abduvakhabov

There are no affiliations available

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