Chemistry of Heterocyclic Compounds

, Volume 14, Issue 1, pp 73–76 | Cite as

Research on benzimidazole derivatives

XLII. Synthesis and transformations of amides of unsaturated carboxylic acids in series of 2-amino derivatives of benzimidazole and pyridine
  • P. V. Tkachenko
  • A. M. Simonov
  • I. I. Popov
Article

Abstract

The acylation of 2-amino derivatives of benzimidazole and pyridine withβ-aryl-α, β-unsaturated carboxylic acid chlorides gave the corresponding amides, which were converted to 2-oxo derivatives of pyrimido [1,2-a]benzimidazole and pyridine by the action of bases.

Keywords

Chloride Organic Chemistry Amide Pyridine Carboxylic Acid 

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Copyright information

© Plenum Publishing Corporation 1978

Authors and Affiliations

  • P. V. Tkachenko
    • 1
  • A. M. Simonov
    • 1
  • I. I. Popov
    • 1
  1. 1.Rostov State UniversityRostov-on-Don

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