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Synthesis and properties of analogs of 5 (or 4)-aminoimidazole-4 (or 5)-carboxamide (AICA) and purines. 13. Synthesis of 5 (or 4)-hydrazinoimidazqles and their derivatives

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

A method for the synthesis of derivatives of 5 (or 4)-hydrazinoimidazole-4 (or 5)-carboxylic acid by reducing the corresponding diazoimidazoles with stannous chloride has been developed, and a number of hydrazones and semicarbazides have been synthesized. It has been shown that under the reduction conditions selected imidazo[4,5-d]-1, 2, 3-triazinone does not have cryptodiazonium properties.

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Authors and Affiliations

  1. S. M. Kirov Ural Polytechnic Institute, 620002, Sverdlovsk

    V. S. Mokrushin, E. F. Golovina, V. I. Nifontov, V. A. Bakulev, T. A. Pospelova & V. K. Usova

Authors
  1. V. S. Mokrushin
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  2. E. F. Golovina
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  3. V. I. Nifontov
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  4. V. A. Bakulev
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  5. T. A. Pospelova
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  6. V. K. Usova
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Additional information

For Report 12, see [1].

Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 11, pp. 1552–1555, November, 1983.

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Mokrushin, V.S., Golovina, E.F., Nifontov, V.I. et al. Synthesis and properties of analogs of 5 (or 4)-aminoimidazole-4 (or 5)-carboxamide (AICA) and purines. 13. Synthesis of 5 (or 4)-hydrazinoimidazqles and their derivatives. Chem Heterocycl Compd 19, 1235–1238 (1983). https://doi.org/10.1007/BF00515367

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  • DOI: https://doi.org/10.1007/BF00515367

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