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Synthesis of 2-acylindoles from α-(N-isatinyl) ketones

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

2-Acylindoles were synthesized by the recyclization of N-phenacyl- and N-aceto-nylisatins in alkaline media and the decarboxylation of 2-acylindolyl-3-carboxylic acids or their salts in basic or neutral media.

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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 11, pp. 1490–1492, November, 1983.

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Gorgos, V.I., Zorin, L.M., Zhungietu, G.I. et al. Synthesis of 2-acylindoles from α-(N-isatinyl) ketones. Chem Heterocycl Compd 19, 1179–1182 (1983). https://doi.org/10.1007/BF00515352

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  • DOI: https://doi.org/10.1007/BF00515352

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