Chemistry of Heterocyclic Compounds

, Volume 17, Issue 2, pp 124–125 | Cite as

Reaction of some benzoxazoline-2-thione derivatives with amines

  • K. Davidkov
  • D. Simov
Article
  • 33 Downloads

Abstract

Hydroxyphenylthioureas were obtained by the reaction of nitro, chloro, bromo, or amino derivatives of benzoxazoline-2-thiones with primary amines. If the substituent in the benzene ring is a nitro group, the reaction with certain secondary amines proceeds with the production of trisubstituted thioureas. It is shown that electron-acceptor substituents in the 5 and 6 positions of the benzene ring facilitate this reaction.

Keywords

Benzene Organic Chemistry Thiourea Chloro Benzene Ring 

Literature cited

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Copyright information

© Plenum Publishing Corporation 1981

Authors and Affiliations

  • K. Davidkov
    • 1
  • D. Simov
    • 1
  1. 1.K. Okhridskii Sofia UniversitySofiaBulgaria

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