Chemistry of Heterocyclic Compounds

, Volume 19, Issue 7, pp 756–762 | Cite as

Synthesis and physicochemical properties of thiazolino[3,2-a]benzimidazoles

  • A. N. Krasovskii
  • N. A. Klyuev
  • A. B. Roman
  • P. M. Kochergin
  • E. Kh. Dank


The reaction of 1-β-hydroxyalkyl(aralkyl)-2-chlorobenzimidazoles with thiourea or the reduction of 1-acylmethylbenzimidazoline-2-thiones with sodium borohydride gave 1-β-hydroxyalkyl(aralkyl, hetaryl)benzimidazoline-2-thiones, which were converted to 2-alkyl(aryl, hetaryl)-substituted thiazolino[3,2-a]benzimidazoles by the action of POCl3.


Sodium Organic Chemistry Physicochemical Property Thiourea Benzimidazole 
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Copyright information

© Plenum Publishing Corporation 1984

Authors and Affiliations

  • A. N. Krasovskii
    • 1
  • N. A. Klyuev
    • 1
  • A. B. Roman
    • 1
  • P. M. Kochergin
    • 1
  • E. Kh. Dank
    • 1
  1. 1.Zaporozhe Medical InstituteZaporozhe

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