Abstract
Substituted 1-pyrimidyl-4-acyl-1,2,3-triazoles were obtained by the reaction of 2- and 4-azidopyrimidines with aryl substituents with acetyl- or benzoylacetone. An accelerating effect of an o-hydroxyphenylpyrimidine fragment in this reaction, which was explained by the effect of an intramolecular hydrogen bond, was observed.
Similar content being viewed by others
Literature cited
V. P. Krivopalov, E. B. Nikolaenkova, V. F. Sedova, and V. P. Mamaev, Khim. Geterotsikl. Soedin., No. 9, 1222 (1983).
T. L. Gilshrist and G. E. Gymer, in: Advances in Heterocyclic Chemistry, A. R. Katritzky and A. J. Boulton, eds., Vol. 16, Academic Press, New York (1974), p. 33.
A. Gorup, M. Kovacic, B. Kranjc-Skraba, B. Mihelcic, S. Simonie, B. Stanovnik, and M. Tisler, Tetrahedron, 30, 2251 (1974).
B. Stanovnik, M. Tisler, S. Polanc, and Ju. Zitnik, Synthesis, No. 7, 491 (1977).
V. V. Solov'eva and É. Yu. Gudrinietse, Khim. Geterotsikl. Soedin., No. 2, 256 (1973).
I. A. Ol'shevskaya, V. Ya. Pochinok, V. V. Kolibaba, and V. I. Rafal'skaya, Vestn. Kievsk. Univ. Khim., 20, 51 (1979).
G. L'Abbe, Ind. Chim. Belge, 34, 519 (1969).
G. Garcia-Munoz, R. Madronero, M. Rico, and M. C. Saldana, J. Heterocycl. Chem., 6, 921 (1969).
O. P. Petrenko, V. P. Krivopalov, V. V. Lapachev, and V. P. Mamaev, Izv. Akad. Nauk SSSR, Ser. Khim., No. 7, 1611 (1980).
O. P. Petrenko, V. P. Krivopalov, V. V. Lapachev, and V. P. Mamaev, Izv. Akad. Nauk SSSR, Ser. Khim., No. 1, 227 (1981).
L. Giammanco and F. P. Invidiata, Atti Accad. Sci., Lett. Arti Palermo, Parte 1, 31, 225 (1972).
Author information
Authors and Affiliations
Additional information
Translated from Khimiya Geterotsiklicheskikh Soedininii, No. 10, pp. 1401–1405, October, 1983.
Rights and permissions
About this article
Cite this article
Krivopalov, V.P., Nikolaenkova, E.B., Sedova, V.F. et al. Reaction of aryl-substituted azidopyrimidines with 1,3-dicarbonyl compounds. Chem Heterocycl Compd 19, 1116–1120 (1983). https://doi.org/10.1007/BF00505770
Received:
Issue Date:
DOI: https://doi.org/10.1007/BF00505770