Skip to main content
Log in

Reaction of aryl-substituted azidopyrimidines with 1,3-dicarbonyl compounds

  • Published:
Chemistry of Heterocyclic Compounds Aims and scope

Abstract

Substituted 1-pyrimidyl-4-acyl-1,2,3-triazoles were obtained by the reaction of 2- and 4-azidopyrimidines with aryl substituents with acetyl- or benzoylacetone. An accelerating effect of an o-hydroxyphenylpyrimidine fragment in this reaction, which was explained by the effect of an intramolecular hydrogen bond, was observed.

This is a preview of subscription content, log in via an institution to check access.

Access this article

Price excludes VAT (USA)
Tax calculation will be finalised during checkout.

Instant access to the full article PDF.

Similar content being viewed by others

Literature cited

  1. V. P. Krivopalov, E. B. Nikolaenkova, V. F. Sedova, and V. P. Mamaev, Khim. Geterotsikl. Soedin., No. 9, 1222 (1983).

    Google Scholar 

  2. T. L. Gilshrist and G. E. Gymer, in: Advances in Heterocyclic Chemistry, A. R. Katritzky and A. J. Boulton, eds., Vol. 16, Academic Press, New York (1974), p. 33.

    Google Scholar 

  3. A. Gorup, M. Kovacic, B. Kranjc-Skraba, B. Mihelcic, S. Simonie, B. Stanovnik, and M. Tisler, Tetrahedron, 30, 2251 (1974).

    Google Scholar 

  4. B. Stanovnik, M. Tisler, S. Polanc, and Ju. Zitnik, Synthesis, No. 7, 491 (1977).

    Google Scholar 

  5. V. V. Solov'eva and É. Yu. Gudrinietse, Khim. Geterotsikl. Soedin., No. 2, 256 (1973).

    Google Scholar 

  6. I. A. Ol'shevskaya, V. Ya. Pochinok, V. V. Kolibaba, and V. I. Rafal'skaya, Vestn. Kievsk. Univ. Khim., 20, 51 (1979).

    Google Scholar 

  7. G. L'Abbe, Ind. Chim. Belge, 34, 519 (1969).

    Google Scholar 

  8. G. Garcia-Munoz, R. Madronero, M. Rico, and M. C. Saldana, J. Heterocycl. Chem., 6, 921 (1969).

    Google Scholar 

  9. O. P. Petrenko, V. P. Krivopalov, V. V. Lapachev, and V. P. Mamaev, Izv. Akad. Nauk SSSR, Ser. Khim., No. 7, 1611 (1980).

    Google Scholar 

  10. O. P. Petrenko, V. P. Krivopalov, V. V. Lapachev, and V. P. Mamaev, Izv. Akad. Nauk SSSR, Ser. Khim., No. 1, 227 (1981).

    Google Scholar 

  11. L. Giammanco and F. P. Invidiata, Atti Accad. Sci., Lett. Arti Palermo, Parte 1, 31, 225 (1972).

    Google Scholar 

Download references

Author information

Authors and Affiliations

Authors

Additional information

Translated from Khimiya Geterotsiklicheskikh Soedininii, No. 10, pp. 1401–1405, October, 1983.

Rights and permissions

Reprints and permissions

About this article

Cite this article

Krivopalov, V.P., Nikolaenkova, E.B., Sedova, V.F. et al. Reaction of aryl-substituted azidopyrimidines with 1,3-dicarbonyl compounds. Chem Heterocycl Compd 19, 1116–1120 (1983). https://doi.org/10.1007/BF00505770

Download citation

  • Received:

  • Issue Date:

  • DOI: https://doi.org/10.1007/BF00505770

Keywords

Navigation