Abstract
The oxidation of N-aminophthalimide with lead tetraacetate in the presence of butenyne and 2-methylbutenyne leads to the corresponding 1-phthalimido-2-ethynylaziridines in good yields.
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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 9, pp. 1176–1178, September, 1991.
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Kuznetsov, M.A., Semenovskii, V.V. & Gindin, V.A. Phthalimidoaziridinylation of the simplest vinylacetylenes. Chem Heterocycl Compd 27, 939–942 (1991). https://doi.org/10.1007/BF00484354
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DOI: https://doi.org/10.1007/BF00484354