Abstract
Reactions between 3-chloroacetylindole and aromatic aldehydes, leading to the formation of the α-oxo epoxides I–IV, have been performed. The reaction of the latter with piperidine and dimethylamine has given α-hydroxy-β-amino ketones of the indole series.
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For Communication LII, see [5].
Translated from Khimiya Geterotsiklicheskikh Soedinenii, Vol. 6, No. 8, pp. 1076–1078, August, 1970.
The authors express their deep gratitude to the Dr. Yu. N. Scheinker and K. F. Turchin for assistance in the interpretation of the PMR spectra.
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Smushkevich, Y.I., Zhigachev, V.E., Sulima, A.V. et al. Indole derivatives. Chem Heterocycl Compd 6, 1004–1006 (1970). https://doi.org/10.1007/BF00480635
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DOI: https://doi.org/10.1007/BF00480635