Chemistry of Heterocyclic Compounds

, Volume 8, Issue 1, pp 46–51 | Cite as

Indole chemistry

XXVIII. 2-oxo-α-carbolines
  • N. N. Borisov
  • R. S. Sagitullin
  • A. N. Kost


The condensation of 1-substituted 2-aminoindoles with β-keto esters gives 2-oxo-α-carbolines. Substitution of diketenes for the β-keto esters leads to a mixture of 2-oxo- and 4-oxo- compounds.


Ester Organic Chemistry Indole Ester Lead Diketenes 
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Copyright information

© Consultants Bureau, a division of Plenum Publishing Corporation 1974

Authors and Affiliations

  • N. N. Borisov
    • 1
  • R. S. Sagitullin
    • 1
  • A. N. Kost
    • 1
  1. 1.M. V. Lomonosov Moscow State UniversityUSSR

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