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Chemistry of Heterocyclic Compounds

, Volume 27, Issue 2, pp 225–227 | Cite as

Reactions of 3-(Β-hydroxyethyl)-8-thiaxanthine

  • é. I. Ivanov
  • A. A. Yavolovskii
  • E. A. Kuklenko
  • O. S. Timofeev
Article
  • 26 Downloads

Abstract

Depending on the base used, reaction of 3-(Β-hydroxyethyl)-8-thiaxanthine with p-toluenesulfonylchloride either stops at the stage of formation of the tosylate or gives 1,2,5-thiadiazolo[3,4-d]oxazolidino[2,3-b]pyrimidin-9(4H)-one. Upon treatment with ammonia or methylamine, both of these compounds react to give 3-(Β-hydroxyethyl)-8-thiaguanines.

Keywords

Ammonia Organic Chemistry Methylamine Tosylate 
These keywords were added by machine and not by the authors. This process is experimental and the keywords may be updated as the learning algorithm improves.

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Copyright information

© Plenum Publishing Corporation 1991

Authors and Affiliations

  • é. I. Ivanov
    • 1
  • A. A. Yavolovskii
    • 1
  • E. A. Kuklenko
    • 1
  • O. S. Timofeev
    • 1
  1. 1.A. V. Bogatskii Physicochemical InstituteAcademy of Sciences of the Ukrainian SSROdessa

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