Abstract
Aminomethylation of pemoline with primary amines has given the corresponding oxazolo[3,2-a]-1,3,5-triazines or oxazolo[3,2-a]-1,3,5,7-tetrazocines. When secondary amines were used, the 5-amino- or 3,5-bis(aminomethyl) derivatives were obtained.
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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 12, pp. 1670–1674, December, 1990.
The authors thank A. V. Dogadin for obtaining and discussing the PMR spectra.
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Ramsh, S.M., Khrabrova, E.S. & Shamina, L.P. Aminomethylation of pemoline. Chem Heterocycl Compd 26, 1387–1391 (1990). https://doi.org/10.1007/BF00473969
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DOI: https://doi.org/10.1007/BF00473969