Abstract
The reaction of 1-acetyl-5-hydroxypyrazolidines with heterocyclic compounds, the amino group of which has an aniline or amidine character, is regioselective and results in the formation of the corresponding hetarylaminopyrazolidines.
Similar content being viewed by others
Literature Cited
L. A. Sviridova, S. V. Afanas'eva, K. N. Zelenin, G. A. Golubeva, I. P. Bezhan, and Yu. G. Bundel', Khim. Geterotsikl. Soed., No. 2, 484 (1987).
K. N. Zelenin, G. A. Golubeva, S. V. Afanas'eva, L. A. Sviridova, I. P. Bezhan, M. Yu. Malov, and Yu. G. Bundel', Khim. Geterotsikl. Soed., No. 9, 1238 (1985).
A. G. Kalandarishvili, P. B. Terent'ev, S. V. Afanas'eva, L. A. Sviridova, R. R. Razakov, Yu. G. Bundel', A. S. Sadykov, and N. S. Kulikov, Khim. Geterotsikl. Soed., No. 10, 1334 (1986).
A. E. Tschitschibabin and E. D. Ossetrova, Berichte, 58, 1708 (1925).
K. S. Sabirov, é. A. Alimov, and S. I. Iskandarov, Paper deposited at VINITI, No. 310–76, February 3, 1976, p. 5; Ref. Zh. Khim., 3Zh341 Dep. (1977).
Ya. L. Gol'dfarb, M. A. Pryanishnikova, and K. A. Zhukova, Izv. Akad. Nauk SSSR, Otd. Khim. Nauk, No. 1, 145 (1953).
G. Joyle and G. Smith, Principles of Chemistry of Heterocyclic Compounds [Russian translation], Mir, Moscow (1975), p. 76.
Author information
Authors and Affiliations
Additional information
Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 9, pp. 1204–1206, September, 1990.
Rights and permissions
About this article
Cite this article
Sviridova, L.A., Golubeva, G.A., Sekhel'meble, V. et al. Reaction of 5-hydroxypyrazolidines with hetarylamines. Chem Heterocycl Compd 26, 1005–1007 (1990). https://doi.org/10.1007/BF00472481
Received:
Issue Date:
DOI: https://doi.org/10.1007/BF00472481