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Indole derivatives.

131. Reaction of 1-acylindoles with acetylchloride and chloroacetylchloride under friedel-crafts conditions

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

Acylation of 1-acylindoles by acetylchloride and chloroacetylchloride in the presence of aluminum chloride leads to formation of 3-acetyl- and 6-chloroacetyl-1-acylindoles, respectively.

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For Communication 130, see [1].

Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 3, pp. 328–330, March, 1989.

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Shner, V.F., Sladkova, T.N., Turchin, K.F. et al. Indole derivatives.. Chem Heterocycl Compd 25, 272–274 (1989). https://doi.org/10.1007/BF00472383

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  • DOI: https://doi.org/10.1007/BF00472383

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