Chemistry of Heterocyclic Compounds

, Volume 5, Issue 3, pp 339–342 | Cite as

Synthesis of derivatives of 5-azabenzofuran with functional substitutes in positions 4 and 7

  • L. N. Yakhontov
  • M. Yu. Uritskaya
  • V. A. Loginova
  • M. V. Rubtsov


Methods for synthesizing derivatives of 5-azabenzofuran with functional substitutes in position 4 and 7 have been elaborated. The reactions of electrophilic substitution in position 7 have been studied.

An examination was made of the substitution of halogens in position 4 of derivatives of 5-azabenzofuran by the methoxy-group during the action of dimethyl sulfate in an aqueous alkali medium.


Sulfate Organic Chemistry Dimethyl Halogen Electrophilic Substitution 
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Copyright information

© Consultants Bureau 1972

Authors and Affiliations

  • L. N. Yakhontov
    • 1
  • M. Yu. Uritskaya
    • 1
  • V. A. Loginova
    • 1
  • M. V. Rubtsov
    • 1
  1. 1.Ordazhonikidze All-Union Scientific-Research Chemical and Pharmaceutical InstituteMoscow

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