Chemistry of Heterocyclic Compounds

, Volume 11, Issue 8, pp 976–978 | Cite as

Synthesis of N-(2-carboxy-4-nitroaryl)-β-alanines and their cyclization to quinoline derivatives

  • A. F. Bekhli
  • L. A. Bolotina


N-(2-Carboxy-4-nitroaryl)-β-alanines were obtained by reaction of 2-chloro-5-nitrobenzoic acids with β-alanine. The products were converted to the corresponding 1,2,3,4-tetrahydro-4-oxo-6-nitroquinolines by cyclization.


Organic Chemistry Quinoline Quinoline Derivative 
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Copyright information

© Plenum Publishing Corporation 1976

Authors and Affiliations

  • A. F. Bekhli
    • 1
  • L. A. Bolotina
    • 1
  1. 1.E. I. Martsinovskii Institute of Medicinal Parasitology and Tropical MedicineMoscow

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