Chemistry of Heterocyclic Compounds

, Volume 14, Issue 10, pp 1085–1087 | Cite as

New methods for the synthesis of amides of benzo[b]thiophene-2carboxylic acid

  • V. L. Savel'ev
  • T. G. Afanas'eva
  • V. A. Zagorevskii


The reaction of 3-bromothiocoumarin with nitrogen bases, during which the thiocoumarin system is converted to a benzothiophene system, was studied. A new method for the synthesis of amides of benzo[b]thiophene-2-carboxylic acid is proposed.


Nitrogen Organic Chemistry Amide Nitrogen Base Benzothiophene 
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Copyright information

© Plenum Publishing Corporation 1979

Authors and Affiliations

  • V. L. Savel'ev
    • 1
  • T. G. Afanas'eva
    • 1
  • V. A. Zagorevskii
    • 1
  1. 1.Scientific-Research Institute of PharmacologyAcademy of Medical Sciences of the USSRMoscow

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