Pharmaceutical Chemistry Journal

, Volume 39, Issue 6, pp 313–315 | Cite as

Synthesis and Antimicrobial Activity of Coordination Compounds of Copper with Substituted Salicylaldehyde Thiosemicarbazones

  • V. I. Prisakar'
  • V. I. Tsapkov
  • S. A. Buracheeva
  • M. S. Byrke
  • A. P. Gulya
Article

Abstract

New coordination compounds of copper(II) with thiosemicarbazones of 5-chloro-, 5-bromo-, 5-nitro-, 5-methyl-, 3,5-dichloro-, and 3,5-dibromo-substituted salicylaldehyde have been synthesized and tested with respect to eight strains of staphyloccoccus, streptococcus, and colon bacillus. These compounds exhibit high antimicrobial activity. The composition and structure of the synthesized complexes have been studied by means of elemental analysis and by magnetochemical, IR, and thermogravimetric techniques. The antimicrobial activity of the obtained coordination compounds depends both on the nature of substituents in the benzene ring of salicylaldehyde and on the nature of acid ligands. The maximum antimicrobial activity was observed for copper(II) complexes with thiosemicarbazone of 3,5-dibromsalicyladehyde.

Keywords

Copper Benzene Organic Chemistry Antimicrobial Activity Benzene Ring 
These keywords were added by machine and not by the authors. This process is experimental and the keywords may be updated as the learning algorithm improves.

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REFERENCES

  1. 1.
    M. D. Mashkovskii, Drugs [in Russian], Belarus, Minsk (1987), Vol. 2, pp. 277–290.Google Scholar
  2. 2.
    G. I. Zhungietu and V. G. Granik, Basic Principles of Drug Design [in Russian], Moldova State University, Chisinau (2000), pp. 264–276.Google Scholar
  3. 3.
    A. B. Tomchin, V. S. Velezheva, and E. B. Shustov, Khim.-Farm. Zh., 32(2), 7–10 (1998).Google Scholar
  4. 4.
    O. V. Fedorova, G. G. Mordovskii, G. L. Rusinov, et al., Khim.-Farm. Zh., 32(2), 11–12 (1998).Google Scholar
  5. 5.
    K. N. Zelenin, O. B. Kuznetsova, A. G. Saminskaya, Khim.-Farm. Zh., 28(2), 34–37 (1994).Google Scholar
  6. 6.
    T. R. Ovsepyan, G. K. Simonyan, G. E. Gabrielyan, et al., Khim.-Farm. Zh., 31(12), 3–5 (1997).Google Scholar
  7. 7.
    T. R. Ovsepyan, G. E. Gabrielyan, G. K. Simonyan, et al., Khim.-Farm. Zh., 34(5), 21–23 (2000).Google Scholar
  8. 8.
    A. V. Ablov and O. A. Bologa, Zh. Neorg. Khim., 19(7), 1964–1968 (1974).Google Scholar
  9. 9.
    A. V. Ablov, N. I. Belichuk, and L. F. Chapurina, Zh. Neorg. Khim., 15(1), 112–118 (1970).Google Scholar
  10. 10.
    N. V. Gerbeleu, Author's Abstract of Cand. Sci. (Chem.) Thesis [in Russian], Moscow (1973).Google Scholar
  11. 11.
    G. N. Pershin, Methods of Experimental Chemotherapy [in Russian], Meditsina, Moscow (1971), pp. 357–359.Google Scholar

Copyright information

© Springer Science+Business Media, Inc. 2005

Authors and Affiliations

  • V. I. Prisakar'
    • 1
  • V. I. Tsapkov
    • 2
  • S. A. Buracheeva
    • 1
  • M. S. Byrke
    • 1
  • A. P. Gulya
    • 2
  1. 1.Moldova State UniversityChisinauMoldova
  2. 2.State University of Medicine and PharmacyChisinauMoldova

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