Advertisement

Springer Nature is making Coronavirus research free. View research | View latest news | Sign up for updates

Synthesis of some aminopropynylpyrazoles

  • 26 Accesses

Conclusions

A number of mono-, di-, and tri(aminopropynyl)pyrazoles was synthesized by the Mannich condensation from pyrazolylacetylenes, and by the condensation of N-substituted propargylamines with iodopyrazoles.

This is a preview of subscription content, log in to check access.

Literature cited

  1. 1.

    G. N. Pershin, S. N. Milovanova, A. L. Mikerina, V. N. Andrievskii, V. E. Aksenova, M. S. Shvartsberg, and I. L. Kotlyarevskii, Izv. Akad. Nauk SSSR, Ser. Khim., 2330 (1969).

  2. 2.

    G. N. Pershin, S. N. Milovanova, A. L. Mikerina, T. G. Shishmakova, M. I. Bardamova, and I. L. Kotlyarevskii, ibid., 1904 (1970).

  3. 3.

    E. G. Izyumov, O. R. Grek, E. K. Andrievskaya, and I. L. Kotlyarevskii, Izv. Sib. Otd. Akad. Nauk SSSR, Ser. Biol. Nauk,1, No. 5, 45 (1969).

  4. 4.

    E. G. Izyumov, P. A. Slabuka, E. K. Andrievskaya, and I. L. Kotlyarevskii, ibid.,2, No. 10, 99 (1969).

  5. 5.

    M. S. Shvartsberg, S. F. Vasilevskii, V. G. Kostrovskii, and I. L. Kotlyarevskii, Khim. Geterotsikl. Soed., 1055 (1969).

  6. 6.

    S. F. Vasilevskii, M. S. Shvartsberg, and I. L. Kotlyarevskii, Izv. Akad. Nauk SSSR, Ser. Khim., 1764 (1971).

  7. 7.

    M. S. Shvartsberg, I. L. Kotlyarevskii, A. N. Kozhevnikova, and V. N. Andrievskii, ibid., 1144 (1970).

  8. 8.

    M. S. Shvartsberg, A. N. Kozhevnikova, and I. L. Kotlyarevskii, ibid., 1833 (1971).

  9. 9.

    G. Papp, L. Szekeres, and T. Szmolenszky, Acta Physiol. Acad. Sci. Hung.,32, 365 (1967).

  10. 10.

    Yu. I. Syrneva, Farmakol. i Toksikol.,17, 27 (1955).

  11. 11.

    Ya. I. Zaidler and A. N. Kudrin, ibid.,28, 662 (1965).

  12. 12.

    R. Huttel, O. Schafer, and P. Jochum, Liebigs Ann. Chem.,593, 200 (1955).

Download references

Author information

Additional information

Translated from Izvestiya Akademii Nauk SSSR, Seriya Khimicheskaya, No. 11, pp. 2524–2529, November, 1972.

Rights and permissions

Reprints and Permissions

About this article

Cite this article

Vasilevskii, S.F., Slabuka, P.A., Izyumov, E.G. et al. Synthesis of some aminopropynylpyrazoles. Russ Chem Bull 21, 2453–2457 (1972). https://doi.org/10.1007/BF00850092

Download citation

Keywords

  • Pyrazole
  • Propargylamines
  • Mannich Condensation
  • Iodopyrazoles