Chemistry of Heterocyclic Compounds

, Volume 21, Issue 2, pp 176–180 | Cite as

Nitrogen-, oxygen-, and sulfur-containing heterocycles. 43. Synthesis and properties of 6-oxo-5H-pyrido[2,3-b][1,4]thiazines

  • N. I. Traven'
  • T. S. Safonova
Article

Abstract

It has previously been observed that the carbamide residue in 2-phenacyl-3-ureido- and 2-cyanomethylpyridine is readily cleaved on cyclization to pyridothiazines [1–4]. It was of interest to establish whether a similar process occurs when the carbonyl component is an α-halo- or unsaturated acid. If this were the case, this reaction could be used to obtain 6-oxopyrido[2,3-b][1,4]thiazines.

Keywords

Oxygen Nitrogen Carbamide Organic Chemistry Carbonyl 
These keywords were added by machine and not by the authors. This process is experimental and the keywords may be updated as the learning algorithm improves.

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Copyright information

© Plenum Publishing Corporation 1985

Authors and Affiliations

  • N. I. Traven'
    • 1
  • T. S. Safonova
    • 1
  1. 1.S. Ordzhonikidze All-Union Scientific Research Institute of Pharmaceutical ChemistryMoscow

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