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Synthesis of Novel Triazolyl-substituted Carboxylic Acid Esters and Their Aminolysis

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Abstract

Recyclization of 4-oxo-1,3-benzoxazinium perchlorates under the action of hydrazinobenzoic acids gave previously unknown 1,2,4-triazolylbenzoic acids which were esterified to obtain the corresponding esters. Alkylation of 3-(o-hydroxyphenyl)-1,2,4-triazoles with ethyl chloroacetate formed ethyl triazolylacetates, whose aminolysis allowed synthesis of novel bis-heterocyclic imides.

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Correspondence to N. I. Vikrishchuk.

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Original Russian Text © N.I. Vikrishchuk, L.D. Popov, 2019, published in Zhurnal Organicheskoi Khimii, 2019, Vol. 55, No. 2, pp. 287–293.

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Vikrishchuk, N.I., Popov, L.D. Synthesis of Novel Triazolyl-substituted Carboxylic Acid Esters and Their Aminolysis. Russ J Org Chem 55, 234–240 (2019). https://doi.org/10.1134/S1070428019020155

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  • DOI: https://doi.org/10.1134/S1070428019020155

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