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Reaction of 2-(nitroamino)pyrimidin-4(3H)-one derivatives with arylamines of low basicity in pivalic acid

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Abstract

Pivalic acid was used as a solvent for aminolysis of poly-substituted 2-(nitroamino)-pyrimidin-4(3Н)-one derivatives with arylamines of low basicity. The reaction did not occur in the other solvents or without solvent. Aminolysis products were obtained in 51–59% yields.

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Authors and Affiliations

  1. Volgograd State Technical University, pr. Lenina 28, Volgograd, 400005, Russia

    I. A. Novakov, A. S. Babushkin, L. L. Brunilina, M. B. Navrotskii, B. S. Orlinson, M. D. Robinovich & A. S. Yablokov

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  1. I. A. Novakov
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  2. A. S. Babushkin
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  3. L. L. Brunilina
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  4. M. B. Navrotskii
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  5. B. S. Orlinson
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  6. M. D. Robinovich
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  7. A. S. Yablokov
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Corresponding author

Correspondence to A. S. Babushkin.

Additional information

Original Russian Text © I.A. Novakov, A.S. Babushkin, L.L. Brunilina, M.B. Navrotskii, B.S. Orlinson, M.D. Robinovich, A.S. Yablokov, 2016, published in Zhurnal Organicheskoi Khimii, 2016, Vol. 52, No. 11, pp. 1659–1661.

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Novakov, I.A., Babushkin, A.S., Brunilina, L.L. et al. Reaction of 2-(nitroamino)pyrimidin-4(3H)-one derivatives with arylamines of low basicity in pivalic acid. Russ J Org Chem 52, 1654–1656 (2016). https://doi.org/10.1134/S1070428016110178

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  • DOI: https://doi.org/10.1134/S1070428016110178

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