3,4,5-Trimethoxy- and 2-, 3-, and 4-acetoxybenzoylglycylglycines and their water-soluble potassium and lithium salts were synthesized. The cerebroprotective properties of the water-soluble potassium and lithium salts of acetoxybenzoylglycylglycines were studied experimentally. The most marked cerebroprotective proteins in cerebral ischemia were found with the lithium salt of 2-acetoxybenzoylglycylglycine.
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Translated from Khimiko-Farmatsevticheskii Zhurnal, Vol. 52, No. 1, pp. 15 – 18, January, 2018.
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Brel’, A.K., Tyurenkov, I.N., Lisina, S.V. et al. Acetoxybenzoylglycylglycines as Potential Cerebroprotective Compounds. Pharm Chem J 52, 37–41 (2018). https://doi.org/10.1007/s11094-018-1762-0
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DOI: https://doi.org/10.1007/s11094-018-1762-0