The reaction of 2-mercaptoimidazoline with 1-iodopropan-2-one or 1,3-diiodopropan-2-one in the absence or in presence of iodine allowed to synthesize new types of annulated heterocyclic systems in one preparative step.
Similar content being viewed by others
References
(а) Yan, K.; Lok, C.-N.; Bierla, K.; Che, C.-M. Chem. Commun. 2010, 46, 7691. (b) Lin, I. W.-S.; Lok, C.-N.; Yan, K.; Che, C.-M. Chem. Commun. 2013, 49, 3297.
Granik, V. G.; Grigor'ev, N. B. Russ. Chem. Bull., Int. Ed. 2002, 51, 1973. [Izv. Akad. Nauk, Ser. Khim. 2002, 1819.]
Johnston, G. A. Clin. Exp. Pharmacol. Physiol. 1992, 19, 73.
Bogatskii, A. V.; Luk'yanenko, N. G.; Kirichenko, T. I. Chem. Heterocycl. Compd. 1983, 19, 577. [Khim. Geterocycl. Soedin. 1983, 723.]
Nomoto, Y.; Obase, H.; Takai, H.; Hirata, T.; Teranishi, M.; Nakamura, J.; Ohno, T.; Kubo, K. Chem. Pharm. Bull. 1990, 38, 2467.
Minch, B. A.; Hickenboth, C. R.; Karabin, R. F.; Zawacky, S. R.; Hockswender, T. R.; McCollum, G. J. US Patent 20090286978.
Kushakova, P. M.; Ramsh, S. M.; Garabadgiu, A. V. Chem. Heterocycl. Compd. 2006, 42, 221. [Khim. Geterocycl. Soedin. 2006, 250.]
Katritzky, A. R.; Wu, J. Synthesis 1994, 597.
Yarosh, N. O.; Zhilitskaya, L. V.; Shagun, L. G.; Dorofeev, I. A. Russ. J. Org. Chem. 2014, 50, 1384. [Zh. Org. Khim. 2014, 1398.]
Silverstein, R. M.; Webster, F. X.; Kiemle, D. J. Spectroscopic Identification of Organic Compounds [Russian translation]; Silverstein, R., Ed.; Binom. Laboratoria Znanii: Moscow, 2011, p. 127.
Reiller, P.; Mercier-Bion, F.; Gimenez, N.; Barre, N.; Miserque, F. Radiochim. Acta 2006, 94, 739.
Shagun, L. G.; Dorofeev, I. A.; Klyba, L.V.; Tokareva, I. A.; Voronkov, M. G. Russ. J. Org. Chem. 2008, 44, 1549. [Zh. Org. Khim. 2008, 44, 1570.]
The main results were obtained by using the instrumentation at Baikal Analytical Center of Collective Use, Siberian Branch of the Russian Academy of Sciences.
Author information
Authors and Affiliations
Corresponding author
Additional information
Translated from Khimiya Geterotsiklicheskikh Soedinenii, 2017, 53(8), 920–923
Rights and permissions
About this article
Cite this article
Shagun, L.G., Dorofeev, I.A., Zhilitskaya, L.V. et al. Synthesis of annulated heterocyclic systems based on 2-mercaptoimidazoline and α-iodo ketones. Chem Heterocycl Comp 53, 920–923 (2017). https://doi.org/10.1007/s10593-017-2146-1
Received:
Accepted:
Published:
Issue Date:
DOI: https://doi.org/10.1007/s10593-017-2146-1