Volume 16, Issue 4, November 2012

ISSN: 1381-1991 (Print) 1573-501X (Online)

In this issue (17 articles)

  1. No Access

    Full-Length Paper

    Combinatorial synthesis of chemical building blocks 1. Azomethines

    Sergey V. Ryabukhin, Dmitriy M. Panov, Andrey S. Plaskon… Pages 625-637
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  2. No Access

    Full-Length Paper

    Synthesis of 2-arylamino substituted 5,6-dihydropyrido[2,3-d]pyrimidine-7(8H)-ones from arylguanidines

    Iñaki Galve, Raimon Puig de la Bellacasa, David Sánchez-García… Pages 639-649
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  3. No Access

    Full-Length Paper

    Tandem synthesis of highly functionalized pyrazole derivatives from terminal alkynes, sulfonyl azides, diethyl azadicarboxylate, and sodium arylsulfinates

    Issa Yavari, Manijeh Nematpour Pages 651-657
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  4. No Access

    Full-Length Paper

    Catalyst-free synthesis of quinazolin-4-ones from (hetero)aryl-guanidines: application to the synthesis of pyrazolo[4,3-f]quinazolin-9-ones, a new family of DYRK1A inhibitors

    Julien Debray, Simon Bonte, Olivier Lozach, Laurent Meijer… Pages 659-667
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  5. No Access

    Full-Length Paper

    CaCl2 as a bifunctional reusable catalyst: diversity-oriented synthesis of 4H-pyran library under ultrasonic irradiation

    Hamid Reza Safaei, Mohsen Shekouhy, Athar Shirinfeshan… Pages 669-683
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  6. No Access

    Full-Length Paper

    A novel microwave synthesis of quinoline-3-carboxylic acid derivatives for treatment against human African trypanosomiasis

    Bhupesh S. Samant, Nyaradzai Nyangari Pages 685-695
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  7. No Access

    Full-Length Paper

    Combretastatin A-4 derivatives: synthesis and evaluation of 2,4,5-triaryl-1H-imidazoles as potential agents against H1299 (non-small cell lung cancer cell)

    Chih-Hua Tseng, Chi-Yi Li, Chien-Chih Chiu, Huei-Ting Hu… Pages 697-709
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  8. No Access

    Full-Length Paper

    Synthesis, crystal structure and biological activity of novel anthranilic diamide insecticide containing alkyl ether group

    Yu Zhao, Li-ping Xu, Jun Tong, Yong-qiang Li, Li-xia Xiong, Fang Li… Pages 711-725
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  9. No Access

    Full-Length Paper

    Synthesis of trans-1,3-diaryl-2-(5-methylisoxazol-3-yl)-2,3-dihydro-1H-naphtho[1,2-e][1,3]oxazines via bismuth(III)-catalyzed one-pot pseudo-four component reaction

    Mehdi Shafiee, Ahmad Reza Khosropour, Iraj Mohammadpoor-Baltork… Pages 727-735
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  10. No Access

    Full-Length Paper

    Synthesis and structure–behavior relationships of tetra-substituted imidazole derivatives of 1,3-diazabicyclo[3,1,0]hex-3-ene

    Nosrat O. Mahmoodi, Manouchehr Mamaghani, Tahereh Behzadi Pages 737-747
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  11. No Access

    Full-Length Paper

    The synthesis of low molecular weight pyrrolo[2,3-c]pyridine-7-one scaffold

    Maxim A. Nechayev, Nikolay Yu. Gorobets, Alexander V. Borisov… Pages 749-757
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  12. No Access

    Full-Length Paper

    GSA: a GPU-accelerated structure similarity algorithm and its application in progressive virtual screening

    Xin Yan, Qiong Gu, Feng Lu, Jiabo Li, Jun Xu Pages 759-769
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  13. No Access

    Full-Length Paper

    A combined 3D-QSAR and molecular docking strategy to understand the binding mechanism of V600EB-RAF inhibitors

    Zaheer Ul-Haq, Uzma Mahmood, Sauleha Reza Pages 771-785
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  14. No Access

    Full-Length Paper

    De novo design of N-(pyridin-4-ylmethyl)aniline derivatives as KDR inhibitors: 3D-QSAR, molecular fragment replacement, protein-ligand interaction fingerprint, and ADMET prediction

    Yanmin Zhang, Haichun Liu, Yu Jiao, Haoliang Yuan, Fengxiao Wang… Pages 787-802
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  15. No Access

    Full-Length Paper

    Molecular docking and receptor-specific 3D-QSAR studies of acetylcholinesterase inhibitors

    Pran Kishore Deb, Anuradha Sharma, Poonam Piplani… Pages 803-823
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  16. No Access

    Full-Length Paper

    Hybridization potential of oligonucleotides comprising 3′-O-methylated altritol nucleosides

    G. Chatelain, G. Schepers, J. Rozenski, Arthur Van Aerschot Pages 825-837
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  17. No Access

    Short Communication

    Synthesis of 3-aryl-1,2,4-benzotriazines via intramolecular cyclization of solid-supported o-hydrazidoanilines

    Edwar Cortés, Luciana Méndez, Ernesto G. Mata, Rodrigo Abonia… Pages 839-846
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