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The Chemistry of Benzotriazole Derivatives pp 1–66Cite as

Preparation, Reactivity, and Synthetic Utility of Simple Benzotriazole Derivatives

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Part of the book series: Topics in Heterocyclic Chemistry ((TOPICS,volume 43))

Abstract

The benzotriazole fragment is known to behave as (1) an excellent leaving group, (2) an electron-donating or an electron-withdrawing group, (3) an anion precursor, and (4) a radical precursor. It confers unique physicochemical properties to its immediate vicinity on various molecular scaffolds. This review covers the preparation and synthetic utility of versatile benzotriazole derivatives. The selected compounds are conveniently prepared from 1H-benzotriazole and are characterized by a huge synthetic potential. Their specific reactivity is discussed and illustrated with various examples ranging from methodology in organic chemistry to the total synthesis of complex structures.

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    Romaric Gérardy & Jean-Christophe M. Monbaliu

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Gérardy, R., Monbaliu, JC.M. (2015). Preparation, Reactivity, and Synthetic Utility of Simple Benzotriazole Derivatives. In: Monbaliu, JC. (eds) The Chemistry of Benzotriazole Derivatives. Topics in Heterocyclic Chemistry, vol 43. Springer, Cham. https://doi.org/10.1007/7081_2015_179

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