Synthesis and Application of (Z)-Alkene- and (E)-Fluoroalkene-Dipeptide Isosteres as cis-Amide Equivalents

Tomita, Kenji; Narumi, Tetsuo; Niida, Ayumu; Oishi, ya; Ohno, Hiroaki; Fujii, Nobutaka

doi:10.1007/978-0-387-73657-0_161

Kenji Tomita⁴,
Tetsuo Narumi⁴,
Ayumu Niida⁴,
ya Oishi⁴,
Hiroaki Ohno⁴ &
…
Nobutaka Fujii⁴

Part of the book series: Advances in Experimental Medicine and Biology ((volume 611))

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References

Niida, A., Tomita, K., Mizumoto, M., Tanigaki, H., Terada, T., Oishi, S., Otaka, A., Inui, K. and Fujii, N. Org. Lett. 8, 613–616 (2006).
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Tomita, K., Niida, A., Oishi, S., Ohno, H., Cluzeau, J., Navenot, J.-M., Wang, Z., Peiper, S. C. and Fujii, N. Bioorg. Med. Chem. 14, 7595–7603 (2006).
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Acknowledgments

We thank Takeda Pharmaceutical Company Limited for the biological activity evaluation of a series of compounds. This work was supported by a Grant-in-Aid for Scientific Research from the Ministry of Education, Culture, Sports, Science, and Technology of Japan, and Health and Labour Sciences Research Grants (Research on HIV/AIDS). K.T., T.N. and A.N. are grateful for Research Fellowships from the JSPS for Young Scientists.

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Authors and Affiliations

Kyoto University Sakyo-ku, Graduate School of Pharmaceutical Sciences, Kyoto, 606-501, Japan
Kenji Tomita, Tetsuo Narumi, Ayumu Niida, ya Oishi, Hiroaki Ohno & Nobutaka Fujii

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Kenji Tomita
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Tetsuo Narumi
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Ayumu Niida
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ya Oishi
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Hiroaki Ohno
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Nobutaka Fujii
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Editors and Affiliations

Department of Chemistry & Biochemistry, New Mexico State University, 1175 N. Horseshoe Drive, Las Cruces, NM, 88003-8001, USA
Susan Del Valle
Department of Pharmacology, University of Sherbrooke Medical School, Sherbrooke, QC, J1H 5N4, Canada
Emanuel Escher
Département de Chimie, Université de Montréal, C.P. 6128, Succursale Centre Ville, Montréal, QC, H3C 3J7, Canada
William D. Lubell

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Tomita, K., Narumi, T., Niida, A., Oishi, y., Ohno, H., Fujii, N. (2009). Synthesis and Application of (Z)-Alkene- and (E)-Fluoroalkene-Dipeptide Isosteres as cis-Amide Equivalents. In: Valle, S.D., Escher, E., Lubell, W.D. (eds) Peptides for Youth. Advances in Experimental Medicine and Biology, vol 611. Springer, New York, NY. https://doi.org/10.1007/978-0-387-73657-0_161

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DOI: https://doi.org/10.1007/978-0-387-73657-0_161
Publisher Name: Springer, New York, NY
Print ISBN: 978-0-387-73656-3
Online ISBN: 978-0-387-73657-0
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