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New methods for the synthesis of amides of benzo[b]thiophene-2carboxylic acid

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

The reaction of 3-bromothiocoumarin with nitrogen bases, during which the thiocoumarin system is converted to a benzothiophene system, was studied. A new method for the synthesis of amides of benzo[b]thiophene-2-carboxylic acid is proposed.

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Authors and Affiliations

  1. Scientific-Research Institute of Pharmacology, Academy of Medical Sciences of the USSR, 125315, Moscow

    V. L. Savel'ev, T. G. Afanas'eva & V. A. Zagorevskii

Authors
  1. V. L. Savel'ev
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  2. T. G. Afanas'eva
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  3. V. A. Zagorevskii
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Additional information

Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 10, pp. 1340–1342, October, 1978.

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Savel'ev, V.L., Afanas'eva, T.G. & Zagorevskii, V.A. New methods for the synthesis of amides of benzo[b]thiophene-2carboxylic acid. Chem Heterocycl Compd 14, 1085–1087 (1978). https://doi.org/10.1007/BF00469946

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  • DOI: https://doi.org/10.1007/BF00469946

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